Original document(11 pages)  中文版
    The invention relates to a method for synthesizing ridge sha tan, which uses the 2-tert-butyl ketonic oxygen amido-3-nitro benzoate (I) and N-(trityl )-5-(4-morphine methylbiphenyll-2-group) tetrazolium (II) as raw material to do N-alkanisation reaction, protecting-released reaction, reduction reaction, ring-closed reaction and ester hydrolytic reaction. <0The protecting-released reaction can slough trityl and tert-butyl ketonic oxygen protect group in the lower aliphatic alcohol organic mixing solution.
Application Number
申请号		 200510131970 Application Date
申请日		 2005.12.22
Title 名称 Method for preparing candestartan
Publication Number
公开号		 1800179 Publication Date
公开日		 2006.07.12
Approval Pub. Date 2007.10.24 Granted Pub. Date 2007.10.24
International Classification 分类号 C07D403/10
Applicant(s) Name
申请人		 Zhejiang Tianyu Pharmaceutical Co., Ltd.
Address 地址
Inventor(s) Name 发明人 Tu Yongjun;Zhang Yi;Cheng Rongde
Attorney & Agent 代理人 ma dongxiao

  
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